Protease Inhibitors and Phosphatase Inhibitors
Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Sumanirole Maleate
An extremely selective dopamine D2 receptor agonist (Ki =
MilliporeSigma™ Calbiochem™ PD 168077 Maleate
A selective D4 dopamine receptor agonist (Ki
MilliporeSigma™ Calbiochem™ (S)-(-)-Raclopride
D2 -like dopamine receptor antagonist targeting D2 R (
MilliporeSigma™ Calbiochem™ (R)-(+)-SKF38393 Hydrochloride
A benzazepine derivative that acts as a selective Dopamine D1 /D5 receptor partial a
MilliporeSigma™ Calbiochem™ (±)-PD 128907 Hydrochloride
Selective dopamine D3 receptor agonist (Ki
MilliporeSigma™ Calbiochem™ (-)-Quinpirole Hydrochloride
A potent, selective dopamine D2 receptor agonist with a Ki valu
MilliporeSigma™ Calbiochem™ SB-277011-A Dihydrochloride
A brain-penetrant, high-affinity, and selective dopamine D3 receptor antagonist
MilliporeSigma™ Calbiochem™ Citalopram Hydrobromide
A potent uptake inhibitor highly selective for 5-HT transporter without effect on noradrenalin or dopamine uptake (IC50
MilliporeSigma™ Calbiochem™ L-741,626
Selective dopamine D2 receptor antagonist that is shown to reversibly block agonist-induced activation of GIRK curre
MilliporeSigma™ Calbiochem™ Bupropion Hydrochloride
Bupropion is a non-selective inhibitor of dopamine and noradrenalin transporters. Also an antagonist for neuronal nicotinic acetylcholine receptors (nAChrs).
MilliporeSigma™ Calbiochem™ GBR 12909 Dihydrochloride
A potent inhibitor of dopamine active transporter (DAT, Ki = 1 nM, IC50 = 40 and 51nM) with >100 fold selectivity over noradrenalin and 5-HT re-uptake trans
Revvity Health Sciences Inc Dopamine D2R expressing cells labeled with Terbium, 200 Tests
Dopaminergic neurons and dopamine receptors are the most numerous in brain. In the brain, dopamine receptors D1 and D2 are GPCR responsible for such crucial processes as voluntary movement, sleep, regulation of food intake, attention, learning, and working memory. Cells expressing the D2 receptor are provided pre-labeled with Terbium, and can be used to conduct receptor binding studies on the aforementioned receptor.
Revvity Health Sciences Inc A1R expressing cells labeled with Terbium, 200 Tests
A1 receptor is one of the four adenosine receptor family (including A2A, A2B and A3 receptors). It has vital role in cardiac and renal processes. It regulates neurotransmitters in the brain, such as dopamine and glutamate. Thus, it is considered as an interesting target in treatment of ischemia-reperfusion injury, renal pathologies, and neuropathic pain. Cells expressing the A1 receptor are provided pre-labeled with Terbium, and can be used to conduct receptor binding studies on the aforementioned receptor.
MilliporeSigma™ Calbiochem™ Dopamine Receptor Antagonist II, Thioridazine, HCl
The Dopamine Receptor Antagonist II, Thioridazine, HCl, also referenced under CAS 130-61-0, controls the biological activity of Dopamine Receptor. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Dopamine Receptor D3 Antagonist II, YQA14
A highly potent and selective antagonist of dopamine D3 receptors. Has two binding sites on human cloned D3 receptors (Ki = 0.0680 pM high affinity and 2.11 nM low affinity).
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