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Tocris Bioscience™ GSK 2606414

Potent and selective PERK inhibitor; orally bioavailable

$442.50 - $1847.00

Specifications

Purity >99%
Product Type GSK 2606414
Molecular Weight (g/mol) 451.44
Inhibitors GSK 2606414
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Products 2
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
51-071-0
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Tocris Bioscience™
5107/10 		10 mg
Each for $442.50
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51-075-0
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Tocris Bioscience™
5107/50 		50 mg
Each for $1,847.00
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Description

Description

Potent and selective protein kinase R-like ER kinase (PERK) inhibitor (IC50 = 0.4 nM). Exhibits >1000-fold selectivity for PERK over HR1 and PKR. Inhibits thapsigargin-induced PERK phosphorylation in lung carcinoma A549 cells. Attenuates subcutaneous pancreatic human tumor xenograft growth in mice. Orally bioavailable.
Specifications

Specifications

>99%
GSK 2606414
451.44
GSK 2606414
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