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  7. GR 125487 sulfamate, Tocris Bioscience™

GR 125487 sulfamate, Tocris Bioscience™

Catalog No. 165850
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

Potent and selective 5-HT4 antagonist; active in vivo

Potent and selective 5-HT4 receptor antagonist (Ki = 0.19 nM for porcine 5-HT4). Centrally active following systemic administration in vivo.

Chemical Identifiers

CAS 859502-43-5
Molecular Formula C19H29FN4O8S2
Molecular Weight (g/mol) 524.579
InChI Key VQJFDBXITIOGJM-UHFFFAOYSA-N
Synonym gr 125487 sulfamate, gr 125487 sulfamate salt, 5-fluoro-2-methoxy-1-2-methylsulfonyl amino ethyl-4-piperidinyl-1h-indole-3-methylcarboxylate sulfamate, tocris-1658, gr-125487 sulfamate salt, 1-2-methanesulfonamido ethyl piperidin-4-yl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate; sulfamic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 5-fluoro-2-methoxy-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, sulfamate 1:1
PubChem CID 6604955
IUPAC Name [1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate;sulfamic acid
SMILES COC1=C(C2=C(N1)C=CC(=C2)F)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C.NS(=O)(=O)O

Specifications

Quantity 50 mg
Formula Weight 524.58
Percent Purity >98%
Chemical Name or Material GR 125487 sulfamate

Safety and Handling

Recommended Storage Desiccate at Room Temperature
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